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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
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/
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85%
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Seq ID
UniProtKB/Swiss-Prot
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Deposition
Contribute data
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UniProt
for
Estrogen receptor beta
Target
Enzymatic
Kinetic
ITC
Articles
Downloads
Primary ID
UniProt Recommended Name
Secondary IDs
BindingDB Name
Ki
IC50
Kd
EC50
k
off
k
on
Lig
Prot
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor [298-554,Y537S]
0
255
0
0
0
0
0
1
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor [298-554,D538G]
0
255
0
0
0
0
0
1
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor [298-554]
0
258
0
0
0
0
0
1
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor [307-554]
0
283
0
0
0
0
0
3
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor [Y537S]
44
218
0
0
0
0
0
3
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor [D538G]
0
251
0
20
0
0
0
2
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor
658
5247
55
1188
0
0
0
342
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estrogen receptor beta
58
356
0
60
0
0
0
36
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
Estradiol-bound Estrogen receptor [255-595]
0
0
5
0
0
0
0
1
P03372
Estrogen receptor
Q13511
Q14276
Q5T5H7
Q6MZQ9
Q9NU51
Q9UDZ7
Q9UIS7
...
760
7123
60
1268
0
0
0
379
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
491
2457
25
782
0
0
0
195
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
Estrogen receptor beta
58
356
0
60
0
0
0
36
Q92731
Estrogen receptor beta
A8K8K5
G3V5M5
O60608
O60685
O60702
O60703
O75583
O75584
Q0MWT5
Q0MWT6
Q86Z31
Q9UEV6
Q9UHD3
Q9UQK9
...
549
2813
25
842
0
0
0
226
2D
3D
TSV